Abstract
Abstract:
The aim of writing this review on gastro retentive and floating drug delivery system was to compile the new literature with the principle mechanism of floatation to acquired gastric retention. Various attempts have been made to develop gastroretentive delivery systems such as high density system, swelling, floating system. In floating multiple unit and single unit system are design and their classification and formulation aspect is cover in detail. These systems are very helpful to different problem solve during the formulation of different dosage form. In this review the gastric physiology and reported intra gastric delivery system have briefly been presented.
References
S. Li et. al., Statistical optimization of gastric floating system for oral controlled delivery of calcium. AAPSPharmSciTech 2001; 2(1) article1.
R. Talukder and R. Fassihi, Gastroretentive Delivery Systems: A mini Review. Drug Development and Industrial Pharmacy 2004; 30(10); 1019-1028.
R. Hejazi and N. Amiji, Stomach specific anti H.Pylori therapy. I: Preparation and characterization of tetracycline of a floating multiple unit capsule, a high density loaded chitosan microspheres. Int. J. Pharm.2002; 235; 87-94.
M P Cooerman, P Krausgrill, K J Hengels, Local gastric and serum amoxicillin concentration after different oral application forms. Antimicrob Agents Chemother1993; 37:1506150g.
B S Dave, A F Amin, M Patel, Gastroretentive drug delivery system of Ranitidine HCl formulation and in vitro evaluation. AAPS PharmSciTech; 2004; 5; 1-10.
W Sawicki, Pharmacokinetics of verapamil and nor verapamil from controlled release floating pellets in humans. Eur J Pharm Biopharm; 2002; 53; 29-35.
B M Singh and K H Kim, Floating drug delivery systems: an approach to oral controlled drug delivery via gastric retention. J Control Release 2000; 63:235-259.
S K Jain, G P Agarwal, N K Jain, Evaluation of porous carrier based floating orlistat microspheres for gastric delivery. AAPS PharmSciTech; 2006:7(4) Article 90.
P Sriamornsak, N Thirawong, S Puttipipatkhachorn, Morphology and buoyancy of oil entrapped calcium pectinate gel beads. The AAPS Journal; 2004; 6(3) Article 24.
J M Patil, R S hirlekar, P S Gide and V J Kadam, Trends in floating drug delivery systems. J SCI IND RES; 2006; 65.
A Rubinstein, Microbially controlled drug delivery to the colon. Biopharm Drug Dispos; 1990; 11; 465-475.
J B Dressman, R R Berardi, L L Dermentzoglou, T L Russell, S P Schmaltz, J L Bernett, K M Jarvenpaa, Upper gastrointestinal pH in seventy nine healthy men and women. Pharm Res; 1990; 7; 756-761.
T L Russell, R R Berardi, J L Bernett, L L Dermentzoglou, K M Jarvenpaa, S P Schmaltz, J B Dressman, Upper gastrointestinal pH in seventy nine healthy elderly North American men and women. Pharm Res; 1993; 10(2); 187-196.
P Mojaverian, H K K Chan (a), Radioelectric determination of gastrointestinal pH in vitro accuracy and in vivo reproducibility in man. Pharm Res; 1998; 5; S-243.
C Y Lui, G L Amidon, R R Berardi, D Fleisher, C Youngberg, J B Dressman. Comparison of gastrointestinal pH in dog and humans: implications on the use of the beagle dog as a model for oral absorption in humans. J Pharm Sci; 1986; 75; 271-274.
S M Shah, J K Patel, N V Patel, Int J Pharm Tech Res; 2009; 1(3); 623-633.
T T Fell, Targeting of drugs and delivery systems to specific sites in the gastrointestinal tract. J Anat; 1996; 189; 517-519.
S K Sarna, Cyclic motor activity: migrating motor complex. Gastroenterology, 1985, 89, 894-913.
M Schemann and J H Ehlein, Mechanical characteristics of phaseII and phase II of the interdigestive migrating motor complex in dogs. Gastroenterology.1986; 91; 117-123.
I R Wilding, A J Coupe, S S Davis. The role of ϒ scintigraphy in oral drug delivery. Adv Drug Deliv Rev; 1991; 7; 87-117.
L Shargel, A Yu, Applied Biopharmaceutics and pharmacokinetics, 4th ed.; Appleton and Lange; Philadelphia, 1999.
A H El-Kamel, M S Sokar, S S Al Gamal, V F Naggar, Preparation and evaluation of ketoprofen floating oral delivery system. Int J Pharm; 2001; 220; 13-21.
S Garg, S Sharma, Gastroretentive drug delivery systems. Business briefing: Pharm Tech; 2003; 160-166.
R Khosla, L C Feely, S S Davis, Gastrointestinal transit of non-disintegrating tablets in fed subjects. Int J Pharm; 1989; 53; 107-17.
C H Kutchai, The gastrointestinal system. In principal of physiology; 2nd Ed.; MR Berna, M N Levy; Eds.; Mosby Year book;St. Louis MO, 1996; 652-686.
S M Reddy, V R Sinha, D S Reddy, Novel and colon-specific drug delivery system for pharmacotherapy of peptide and non-peptide drugs. Drugs Today; 1999; 35(7); 537-580.
P Mojaverian, P H Vlasses, P E Kellner, M L Rocci. Effect of gender, posture and age on gastric residence time of an indigestible solid: Pharmaceutical considerations. Pharm Res; 1998; 5(10); 639-643.
S S Davis, R Khosla, C G Wilson, N Washington, The
gastrointestinal transit of a controlled release pellet formulation of tiaprofemic acid. Int J Pharm; 1987; 33; 253-258.
R Kinget, W Kalala, L Vervoort, G V Mooter, Colonic drug targeting. J Drug Target; 1998; 6(2), 129-149.
H M Park, J M Cherish, B D Rosenback, R L Brunelle, B Hargrove, H N Wellman, Gastric emptying of enteric-coated tablets. Dig Dis Sci; 1984; 29; 207-212.
Y Kawashima, T Niwa, H Takeuchi H, T Hino, Y Itoh. J Pharm Sci; 1996; 4; S182.
A Rubinstein, D R Friend. Specific delivery to the gastrointestinal tract. In Domb AJ (Ed) polymeric site specific pharmacotherapy, wiley; Chichester; 1994; pp 282-283.
W A Ritschel, Targeting in the gastrointestinal tract: new approaches, methods, Find Exp Clin Pharmacol, 13(1991) 313-336.
A S Michaels, Drug delivery device with self actuated mechanism for retaining device in selected area. US pat 3; 786; 813; January 22, 1974.
H Hasim and Po A Li Wan, Improving the release characteristics of water-soluble drug from hydrophilic sustained release matrices by in situ gas-generation. Int J Pharm; 35; 1987; 201-206.
M Ichikawa, S Watanabe, Y Miyake, A new multiple unit oral floating dosage system, I: Preparation and in vitro evaluation of floating and sustained release kinetics. J Pharm Sci; 1991; 80; 1062-1066.
F Atyabi, H L Sharma, A H Mahannad, J T Fell, In vivo evaluation of a novel gastric retentive formulation based on ion exchange resins. J Control release; 42(1996); 105-113.
R B Umamaheshwari, S Jain, N K Jain, A new approach in gastroretentive drug delivery system using cholestyramine; Drug Deliv; 10; 2003; 151-160.
L Yang, J Esharghi, R Fassihi, A new intra gastric delivery system for the treatment of Helicobacter Pylori associated gastric ulcers: in vitro evaluation. J Control Release; 1999; 57; 215-222.
A S Michael, J D Bishaw, A Zaffaroni, Gastro inflatable drug delivery device. US Pat 3; 901; 232; 1975.
I Krogel and R Bodomeier, Floating or pulsatile drug delivery systems based on coated effervescent cores. Int J Pharm; 187; 1999; 175-184.
P R Sheth, J L Tossounian J L, Sustained release pharmaceutical capsules. US Pat 4; 126; 672; November 21, 1978.
S Desai and S Bolton, A controlled release drug delivery system: In vitro- in vivo evaluation. Pharm Res; 10; 1993; 1321-1325.
P Dennis, K Timmins, S Lee, Buoyant controlled release powder formulation. US Pat 5; 169; 638; December 8, 1992.
R M Harrigan, Drug delivery device for preventing contact of undissolved drug with the stomach lining. US Pat 4, 055; 178; October 25, 1977.
J H Lee, T G Park, Y B Lee, S C Shin, H H Choi, effect of adding non volatile oil as a core material for the floating microsphere prepared by emulsion solvent diffusion method. J Microencapsulation; 2001; 18; 65-75.
Y D Tong, S S Venkatraman, F Y C Boey, Li-Wei Wong, Sustained release of hydrophobic and hydrophilic drugs from a floating dosage form. Int J Pharm; 336; 2007; 159-165.
J Timmermans, J M Andre, Factors controlling the buoyancy and gastric retention capabilities of floating matrix capsules: new data for reconsidering the controversy. J Pharm Sci; 1994; 83; 18-24.
A Streubel, J Siepmann, R Bodomeier, Floating microparticles based on low-density foam powder. Int J Pharm; 241; 2002; 279-292.
B V Gansbeke, J Timmermans, A Schoutens, A J Moes, Intra gastric positioning of two concurrently ingested pharmaceutical matrix dosage forms. Nucl Med Biol; 18; 1991; 711-718.
R E Horton, FGM Ross, G H Darling, Determination of the emptying time of the stomach by use of enteric coated barium granules. Br Med J; 1; 1965; 1537-1539.
F Jwo, D E Edgren, P S Wong, Gastric retention dosage forms having multiple layers. Int Applications W00038650; July6, 2000.
W R Hendee, Textbook of Diagnostic imaging II, Vol.I, edited by C E Putman and C E Ravin (W B Saunders, Philadelphia) 1994, 1-6.
A Steingotter, D Weishaupt, P Kunz Meda, K Legsfeld, H M Thumshirn, P Boesinger, M Fried, W Schwizer, Magnetic resonance imaging for the in vivo evaluation of gastric retentive tablets. Pharm Res; 2003; 20; 2001-2007.
L Shoufeng, L Senshang, P D Bruce, L H Mirchandani, Y W Chien, Effect of formulation variables on the floating properties of gastric floating drug delivery system. Drug Dev Ind Pharm; 2000; 28(7); 783-793.
V F Patel and N M Patel, Intra gastric floating drug delivery system of cefuroxime Axetil: In vitro evaluation. AAPS PharmSciTech; 2006; 7(1); Article 17.
D M Patel, N M Patel, N M Pandya, P D Jogani, Formulation and optimization of carbamazepine floating tablets. Ind J Pharm Sci; 2007; 69(6); 763-767.
C Narendra, M S Srinath, Ganesh Babu, Optimization of bilayer floating tablets containing metoprolol tartrate as a model drug for gastric retention. AAPS PharmSciTech; 2006; 7(2); Article 34.
S Sharma, P Atmaram, Low-density multiparticulate system for pulsatile release of meloxicam. Int J Pharm; 2006; 313; 150-158.
S Sungthongjeen, P Ornlakasana, Limmatvapirat, Puttipipatkhachorn, Preparation and in vitro evaluation of multiple unit floating drug delivery system based on gas formation technique. Int J Pharm; 2006; 324; 136-143.
R D Kale, P T tayade. A multiple unit floating drug delivery system of piroxiacm using eudragit polymer. Ind J Pharm Sci; 200769(1); 120-123.
P R Nepal, M K Chun, H K Choi. Preparartion of floating microspheres for fish farming. Int J Pharm; 2007; 341; 85-90.
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